Ibudilast, also known as AV411 or MN-166, is a potent phosphodiesterase (PDE) inhibitor and neuroprotective agent, used in the treatment of neurological diseases, chronic pain, opioid withdrawal, and multiple sclerosis (MS). With anti-inflammatory and glial cell modulating properties, Ibudilast is gaining increased attention in neuropharmacology and addiction medicine.
At Yikang Chemical, we supply high-purity Ibudilast suitable for pharmaceutical R&D, formulation development, and advanced CNS drug research.
✅ Product Specifications – Ibudilast
- Product Name: Ibudilast
- CAS Number: 50847-11-5
- Molecular Formula: C14H18N2O
- Molecular Weight: 230.31 g/mol
- Appearance: White to off-white crystalline powder
- Purity: ≥99% (HPLC)
- Synonyms: AV411, MN-166, KC-404, 3-Isobutyryl-2-isopropylpyrazolo[1,5-a]pyridine
🧪 Applications & Therapeutic Uses
- Neuroprotective treatment for Multiple Sclerosis (MS), ALS, stroke
- Chronic neuropathic pain management
- Adjunct therapy for opioid withdrawal and addiction
- Clinical trials in depression, alcoholism, and neuroinflammation
Ibudilast acts by inhibiting PDE4 and PDE10, and modulating glial cell activation, reducing pro-inflammatory cytokine release in the CNS, thereby improving neuronal survival and reducing neurodegeneration.
🏭 Why Choose Yikang Chemical?
- ✅ ≥99% HPLC Purity – Suitable for R&D and formulation testing
- ✅ Technical Documentation – COA, MSDS, NMR, and route of synthesis available
- ✅ Custom Synthesis & Bulk Supply – Flexible scale: mg to kg
- ✅ Fast Delivery – Global logistics and export support
- ✅ Consistent Quality – Strict QC, low impurities, GMP-like conditions
Whether for clinical research, pre-clinical studies, or API scale-up, our Ibudilast is widely adopted by CROs, pharmaceutical companies, and university labs worldwide.
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📦 Packaging & Logistics
- Standard Packaging: Aluminum foil bag / HDPE drum
- MOQ: 100g for lab R&D; bulk quantities available
- Labeling: GHS-compliant with batch traceability
- Storage: Keep sealed in cool, dry place; protect from light
- Shipping: FedEx, DHL, air/sea freight with full export documentation
📞 Contact Us for Quote, Sample, or Technical Sheet
Looking for a trusted supplier of Ibudilast (CAS 50847-11-5) with fast lead times and solid quality assurance? Yikang Chemical provides tailored solutions for your R&D and commercial needs.
🌐 Website: www.yikanghuagong.com
📧 Email: yikangmelody@163.com